5X72
The crystal Structure PDE delta in complex with (rac)-p9
Functional Information from GO Data
Chain | GOid | namespace | contents |
A | 0005095 | molecular_function | GTPase inhibitor activity |
A | 0005515 | molecular_function | protein binding |
A | 0005737 | cellular_component | cytoplasm |
A | 0005829 | cellular_component | cytosol |
A | 0005856 | cellular_component | cytoskeleton |
A | 0005929 | cellular_component | cilium |
A | 0007601 | biological_process | visual perception |
A | 0016020 | cellular_component | membrane |
A | 0030659 | cellular_component | cytoplasmic vesicle membrane |
A | 0031267 | molecular_function | small GTPase binding |
A | 0031410 | cellular_component | cytoplasmic vesicle |
A | 0042995 | cellular_component | cell projection |
A | 0050953 | biological_process | sensory perception of light stimulus |
Functional Information from PDB Data
site_id | AC1 |
Number of Residues | 11 |
Details | binding site for residue P59 A 201 |
Chain | Residue |
A | LEU17 |
A | P69202 |
A | HOH331 |
A | MET20 |
A | TRP32 |
A | ARG61 |
A | GLN78 |
A | ILE109 |
A | THR131 |
A | VAL145 |
A | LEU147 |
site_id | AC2 |
Number of Residues | 9 |
Details | binding site for residue P69 A 202 |
Chain | Residue |
A | LEU22 |
A | ILE53 |
A | LEU54 |
A | TRP90 |
A | ILE109 |
A | SER115 |
A | GLN116 |
A | TYR149 |
A | P59201 |