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5WPB

Crystal structure of fragment 3-(3-(pyridin-2-ylmethoxy)quinoxalin-2-yl)propanoic acid bound in the ubiquitin binding pocket of the HDAC6 zinc-finger domain

Functional Information from GO Data
ChainGOidnamespacecontents
A0008270molecular_functionzinc ion binding
Functional Information from PDB Data
site_idAC1
Number of Residues4
Detailsbinding site for residue ZN A 1301
ChainResidue
ACYS1145
ACYS1148
AHIS1164
AHIS1170

site_idAC2
Number of Residues4
Detailsbinding site for residue ZN A 1302
ChainResidue
ACYS1133
ACYS1136
ACYS1153
AHIS1160

site_idAC3
Number of Residues4
Detailsbinding site for residue ZN A 1303
ChainResidue
AHIS1115
ACYS1183
ACYS1186
ACYS1113

site_idAC4
Number of Residues16
Detailsbinding site for residue B8P A 1304
ChainResidue
AGLU1141
ATRP1143
AGLY1154
AARG1155
ATYR1156
ASER1175
AASP1178
ASER1180
ATRP1182
ATYR1184
ATYR1189
AASN1200
AHIS1203
AHOH1409
AHOH1411
AHOH1467

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues6
DetailsMOD_RES: Phosphothreonine => ECO:0007744|PubMed:24275569
ChainResidueDetails
ASER1168
AVAL1173
ALEU1179
ACYS1183
ACYS1186
AHIS1192

site_idSWS_FT_FI2
Number of Residues1
DetailsMOD_RES: Phosphoserine => ECO:0007744|PubMed:24275569
ChainResidueDetails
AGLN1187

222415

PDB entries from 2024-07-10

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