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5WMG

N-terminal bromodomain of BRD4 in complex with OTX-015

Functional Information from PDB Data
site_idAC1
Number of Residues6
Detailsbinding site for residue EDO A 201
ChainResidue
A6JF204
AHOH302
AHOH308
AHOH344
AHOH398
AHOH512

site_idAC2
Number of Residues9
Detailsbinding site for residue EDO A 202
ChainResidue
AALA122
AGLU167
AHOH362
AHOH382
AHOH409
AHOH426
AGLU49
AGLN62
AASN121

site_idAC3
Number of Residues7
Detailsbinding site for residue EDO A 203
ChainResidue
AILE100
AILE101
ALYS102
ATHR103
AASN135
AASP145
AHOH301

site_idAC4
Number of Residues17
Detailsbinding site for residue 6JF A 204
ChainResidue
ATRP81
APRO82
APHE83
AGLN85
ALYS91
ALEU92
AASN140
AASP145
AMET149
AEDO201
AHOH310
AHOH314
AHOH316
AHOH321
AHOH420
AHOH529
AHOH564

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues1
DetailsSITE: Acetylated histone binding => ECO:0000269|PubMed:22464331
ChainResidueDetails
AASN140

site_idSWS_FT_FI2
Number of Residues2
DetailsCROSSLNK: Glycyl lysine isopeptide (Lys-Gly) (interchain with G-Cter in SUMO2) => ECO:0007744|PubMed:28112733
ChainResidueDetails
ALYS99

225399

PDB entries from 2024-09-25

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