5WMD
N-terminal bromodomain of BRD4 in complex with OTX-015
Functional Information from PDB Data
site_id | AC1 |
Number of Residues | 13 |
Details | binding site for residue 6JE A 201 |
Chain | Residue |
A | PRO53 |
A | MET149 |
A | HOH306 |
A | HOH330 |
A | HOH374 |
A | TRP81 |
A | PRO82 |
A | LEU92 |
A | LEU94 |
A | LYS99 |
A | LYS102 |
A | ASN140 |
A | ILE146 |
Functional Information from SwissProt/UniProt
site_id | SWS_FT_FI1 |
Number of Residues | 1 |
Details | SITE: Acetylated histone binding => ECO:0000269|PubMed:22464331 |
Chain | Residue | Details |
A | ASN140 |
site_id | SWS_FT_FI2 |
Number of Residues | 2 |
Details | CROSSLNK: Glycyl lysine isopeptide (Lys-Gly) (interchain with G-Cter in SUMO2) => ECO:0007744|PubMed:28112733 |
Chain | Residue | Details |
A | LYS99 |