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5WKM

2.25 A resolution structure of MERS 3CL protease in complex with piperidine-based peptidomimetic inhibitor 21

Functional Information from GO Data
ChainGOidnamespacecontents
A0008233molecular_functionpeptidase activity
A0019082biological_processviral protein processing
Functional Information from PDB Data
site_idAC1
Number of Residues12
Detailsbinding site for residue N02 A 401
ChainResidue
APHE143
AASP190
AB6Y402
AHOH534
AGLY146
ASER147
ACYS148
AHIS166
AGLN167
AMET168
AGLU169
AHIS175

site_idAC2
Number of Residues12
Detailsbinding site for residue B6Y A 402
ChainResidue
AHIS41
APHE143
ASER147
ACYS148
AHIS166
AGLN167
AMET168
AGLU169
AHIS175
AASP190
AN02401
AHOH534

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues2
DetailsActive site: {"description":"For 3CL-PRO activity","evidences":[{"source":"PROSITE-ProRule","id":"PRU00772","evidenceCode":"ECO:0000255"}]}
ChainResidueDetails

246704

PDB entries from 2025-12-24

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