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5WKL

1.85 A resolution structure of MERS 3CL protease in complex with piperidine-based peptidomimetic inhibitor 17

Functional Information from GO Data
ChainGOidnamespacecontents
A0008233molecular_functionpeptidase activity
A0019082biological_processviral protein processing
Functional Information from PDB Data
site_idAC1
Number of Residues15
Detailsbinding site for residue AVY A 401
ChainResidue
AHIS41
AGLU169
AHIS175
AASP190
AGLN192
AB3J402
AHOH564
ATHR62
AHIS64
APHE143
ACYS145
ACYS148
AHIS166
AGLN167
AMET168

site_idAC2
Number of Residues16
Detailsbinding site for residue B3J A 402
ChainResidue
ATHR62
AHIS64
APHE143
ACYS145
AGLY146
ASER147
ACYS148
AHIS166
AGLN167
AMET168
AGLU169
AHIS175
AASP190
AGLN192
AAVY401
AHOH564

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues2
DetailsActive site: {"description":"For 3CL-PRO activity","evidences":[{"source":"PROSITE-ProRule","id":"PRU00772","evidenceCode":"ECO:0000255"}]}
ChainResidueDetails

248335

PDB entries from 2026-01-28

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