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5WKJ

2.05 A resolution structure of MERS 3CL protease in complex with inhibitor GC376

Functional Information from GO Data
ChainGOidnamespacecontents
A0008233molecular_functionpeptidase activity
A0019082biological_processviral protein processing
Functional Information from PDB Data
site_idAC1
Number of Residues5
Detailsbinding site for residue CA A 401
ChainResidue
AHOH504
AHOH554
AHOH564
AHOH587
AHOH662

site_idAC2
Number of Residues5
Detailsbinding site for residue CA A 402
ChainResidue
AHOH668
ATHR101
AHOH589
AHOH629
AHOH652

site_idAC3
Number of Residues15
Detailsbinding site for residue B1S A 403
ChainResidue
AHIS41
AHIS64
APHE143
ALEU144
ACYS145
ACYS148
AHIS166
AGLN167
AMET168
AGLU169
AHIS175
AASP190
AGLN192
AK36404
AHOH580

site_idAC4
Number of Residues15
Detailsbinding site for residue K36 A 404
ChainResidue
AHIS64
APHE143
ALEU144
ACYS145
AGLY146
ASER147
ACYS148
AHIS166
AGLN167
AMET168
AGLU169
AHIS175
AGLN192
AB1S403
AHOH580

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues2
DetailsACT_SITE: For 3CL-PRO activity => ECO:0000255|PROSITE-ProRule:PRU00772
ChainResidueDetails
AHIS41
ACYS148

site_idSWS_FT_FI2
Number of Residues1
DetailsSITE: Cleavage; by 3CL-PRO => ECO:0000250
ChainResidueDetails
AGLN306

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PDB entries from 2024-07-10

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