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5WIM

JAK2 Pseudokinase in complex with AT9283

Functional Information from GO Data
ChainGOidnamespacecontents
A0004672molecular_functionprotein kinase activity
A0005524molecular_functionATP binding
A0006468biological_processprotein phosphorylation
Functional Information from PDB Data
site_idAC1
Number of Residues12
Detailsbinding site for residue 35R A 901
ChainResidue
ALEU551
AASN678
ALEU680
ASER698
ALEU579
ALYS581
AGLU627
AVAL629
ALYS630
APHE631
AGLY632
ALYS677

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues1
DetailsSITE: Breakpoint for translocation to form PCM1-JAK2 fusion protein
ChainResidueDetails
AASP710

site_idSWS_FT_FI2
Number of Residues1
DetailsMOD_RES: Phosphotyrosine => ECO:0007744|PubMed:23186163
ChainResidueDetails
ATYR570

218853

PDB entries from 2024-04-24

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