Loading
PDBj
MenuPDBj@FacebookPDBj@TwitterPDBj@YouTubewwPDB FoundationwwPDB
RCSB PDBPDBeBMRBAdv. SearchSearch help

5W0Q

CREBBP Bromodomain in complex with Cpd17 (N,2,7-trimethyl-2,3-dihydro-4H-benzo[b][1,4]oxazine-4-carboxamide)

Functional Information from GO Data
ChainGOidnamespacecontents
A0004402molecular_functionhistone acetyltransferase activity
A0006355biological_processregulation of DNA-templated transcription
Functional Information from PDB Data
site_idAC1
Number of Residues3
Detailsbinding site for residue SO4 A 1201
ChainResidue
AARG1112
AARG1112
AHOH1386

site_idAC2
Number of Residues4
Detailsbinding site for residue SO4 A 1202
ChainResidue
AARG1169
AARG1169
AHOH1347
AHOH1347

site_idAC3
Number of Residues3
Detailsbinding site for residue SO4 A 1203
ChainResidue
AHOH1301
ASER1172
AARG1173

site_idAC4
Number of Residues6
Detailsbinding site for residue 9UG A 1204
ChainResidue
APRO1110
APHE1111
ALEU1119
AASN1168
AHOH1309
AHOH1365

Functional Information from PROSITE/UniProt
site_idPS00633
Number of Residues60
DetailsBROMODOMAIN_1 Bromodomain signature. SlpFrqpvDpqllgipDYFdiVknpMdlstIkrkldtgq..Yqepwqyvddvwl.MfnNAwlY
ChainResidueDetails
ASER1108-TYR1167

222624

PDB entries from 2024-07-17

PDB statisticsPDBj update infoContact PDBjnumon