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5VQT

Crystal Structure of HIV-1 Reverse Transcriptase in Complex with 2-chloro-N-(6-cyano-3-(2-(2-(2,4-dioxo-3,4-dihydropyrimidin-1(2H)-yl)ethoxy)phenoxy)-4-methylnaphthalen-1-yl)-N-methylacetamide (JLJ686), a Non-nucleoside Inhibitor

Functional Information from GO Data
ChainGOidnamespacecontents
A0003676molecular_functionnucleic acid binding
A0003964molecular_functionRNA-directed DNA polymerase activity
A0004523molecular_functionRNA-DNA hybrid ribonuclease activity
A0006278biological_processRNA-templated DNA biosynthetic process
B0003964molecular_functionRNA-directed DNA polymerase activity
B0006278biological_processRNA-templated DNA biosynthetic process
Functional Information from PDB Data
site_idAC1
Number of Residues15
Detailsbinding site for residue 9K7 A 601
ChainResidue
APRO95
AGLY190
APHE227
ATRP229
AHIS235
APRO236
ATYR318
ALYS101
ALYS102
ALYS103
AVAL106
AVAL179
ATYR181
ATYR183
ATYR188

site_idAC2
Number of Residues4
Detailsbinding site for residue SO4 A 602
ChainResidue
AARG277
AARG356
AMET357
AARG358

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues8
DetailsRegion: {"description":"RT 'primer grip'"}
ChainResidueDetails

site_idSWS_FT_FI2
Number of Residues32
DetailsMotif: {"description":"Tryptophan repeat motif"}
ChainResidueDetails

site_idSWS_FT_FI3
Number of Residues6
DetailsBinding site: {}
ChainResidueDetails

site_idSWS_FT_FI4
Number of Residues4
DetailsBinding site: {"evidences":[{"evidenceCode":"ECO:0000305"}]}
ChainResidueDetails

site_idSWS_FT_FI5
Number of Residues4
DetailsSite: {"description":"Essential for RT p66/p51 heterodimerization"}
ChainResidueDetails

site_idSWS_FT_FI6
Number of Residues1
DetailsSite: {"description":"Cleavage; by viral protease; partial"}
ChainResidueDetails

239149

PDB entries from 2025-07-23

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