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5VB6

X-ray co-structure of nuclear receptor ROR-gammat Ligand Binding Domain with an inverse agonist and SRC2 peptide

Functional Information from GO Data
ChainGOidnamespacecontents
A0003677molecular_functionDNA binding
A0004879molecular_functionnuclear receptor activity
A0005634cellular_componentnucleus
A0006355biological_processregulation of DNA-templated transcription
Functional Information from PDB Data
site_idAC1
Number of Residues5
Detailsbinding site for residue NA A 601
ChainResidue
ACYS366
ATYR369
ASER408
AHOH794
AHOH828

site_idAC2
Number of Residues17
Detailsbinding site for residue 927 A 602
ChainResidue
AHIS323
ALEU324
AVAL361
AARG364
AMET365
AARG367
APHE388
ALEU396
APHE401
AHIS479
ATYR502
AHOH769
AHOH826
ACYS285
AGLN286
ATRP317
ACYS320

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues5
DetailsMotif: {"description":"AF-2"}
ChainResidueDetails

site_idSWS_FT_FI2
Number of Residues4
DetailsMotif: {"description":"LXXLL motif 2"}
ChainResidueDetails

239803

PDB entries from 2025-08-06

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