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5V5D

Room temperature (280K) crystal structure of Kaposi's sarcoma-associated herpesvirus protease in complex with allosteric inhibitor (compound 250)

Functional Information from GO Data
ChainGOidnamespacecontents
A0004252molecular_functionserine-type endopeptidase activity
A0006508biological_processproteolysis
B0004252molecular_functionserine-type endopeptidase activity
B0006508biological_processproteolysis
Functional Information from PDB Data
site_idAC1
Number of Residues7
Detailsbinding site for residue 8OY A 201
ChainResidue
AILE105
ATRP109
AHOH337
BLEU47
BPRO192
B8OY201
B8OY202

site_idAC2
Number of Residues12
Detailsbinding site for residue 8OY B 201
ChainResidue
BLEU79
BLEU83
BVAL89
BTRP109
BSER191
BPRO192
BLEU193
BGLU194
BTHR195
BHOH317
ATRP109
A8OY201

site_idAC3
Number of Residues10
Detailsbinding site for residue 8OY B 202
ChainResidue
AARG82
ALEU83
ASER87
ATRP109
A8OY201
BILE44
BALA139
BLEU140
BHOH308
BHOH338

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PDB entries from 2024-07-10

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