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5UT4

JAK2 JH2 in complex with NVP-BSK805

Functional Information from GO Data
ChainGOidnamespacecontents
A0004672molecular_functionprotein kinase activity
A0005524molecular_functionATP binding
A0006468biological_processprotein phosphorylation
Functional Information from PDB Data
site_idAC1
Number of Residues15
Detailsbinding site for residue DQX A 901
ChainResidue
ALEU551
ASER633
ATHR636
ALYS677
ALEU680
ASER698
AHOH1057
AILE559
ALEU579
AGLU627
APHE628
AVAL629
ALYS630
APHE631
AGLY632

site_idAC2
Number of Residues5
Detailsbinding site for residue GOL A 902
ChainResidue
AASN673
AARG715
ATRP718
AHOH1049
AHOH1050

site_idAC3
Number of Residues2
Detailsbinding site for residue GOL A 903
ChainResidue
AILE682
AARG683

site_idAC4
Number of Residues3
Detailsbinding site for residue DMS A 904
ChainResidue
AALA774
AALA781
AASN782

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues1
DetailsSITE: Breakpoint for translocation to form PCM1-JAK2 fusion protein
ChainResidueDetails
AASP710

site_idSWS_FT_FI2
Number of Residues1
DetailsMOD_RES: Phosphotyrosine => ECO:0007744|PubMed:23186163
ChainResidueDetails
ATYR570

222624

PDB entries from 2024-07-17

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