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5UT1

JAK2 JH2 in complex with BI-D1870

Functional Information from GO Data
ChainGOidnamespacecontents
A0004672molecular_functionprotein kinase activity
A0005524molecular_functionATP binding
A0006468biological_processprotein phosphorylation
Functional Information from PDB Data
site_idAC1
Number of Residues6
Detailsbinding site for residue GOL A 901
ChainResidue
AASN673
ACYS675
AARG715
ATRP718
AGOL902
AHOH1067

site_idAC2
Number of Residues10
Detailsbinding site for residue GOL A 902
ChainResidue
ALYS677
AASN678
AARG715
AGOL901
AHOH1005
AHOH1018
AHOH1092
AGLY554
ATHR555
AASN673

site_idAC3
Number of Residues6
Detailsbinding site for residue GOL A 903
ChainResidue
AARG588
AVAL617
AGLY619
AASP620
AGLU621
AASN622

site_idAC4
Number of Residues4
Detailsbinding site for residue GOL A 904
ChainResidue
AHIS606
AHOH1007
AHOH1020
AHOH1183

site_idAC5
Number of Residues15
Detailsbinding site for residue 7DZ A 905
ChainResidue
ALEU551
ALEU579
ALYS581
AVAL610
AGLN626
AGLU627
APHE628
AVAL629
AGLY632
ALYS677
ALEU680
ASER698
AHOH1049
AHOH1092
AHOH1107

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues1
DetailsSITE: Breakpoint for translocation to form PCM1-JAK2 fusion protein
ChainResidueDetails
AASP710

site_idSWS_FT_FI2
Number of Residues1
DetailsMOD_RES: Phosphotyrosine => ECO:0007744|PubMed:23186163
ChainResidueDetails
ATYR570

221051

PDB entries from 2024-06-12

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