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5PAK

Crystal Structure of Factor VIIa in complex with N-[[4-(aminomethyl)-2-(2-amino-2-oxoethoxy)phenyl]methyl]-2-(4-hydroxyphenyl)-2-methoxyacetamide;hydrochloride

Functional Information from GO Data
ChainGOidnamespacecontents
C0004252molecular_functionserine-type endopeptidase activity
C0006508biological_processproteolysis
Functional Information from PDB Data
site_idAC1
Number of Residues6
Detailsbinding site for residue CA C 501
ChainResidue
CGLU270
CASP272
CGLU275
CGLU280
CHOH650
CHOH798

site_idAC2
Number of Residues7
Detailsbinding site for residue SO4 C 502
ChainResidue
CHOH632
CHOH670
CHOH679
CHOH765
CMET366
CTHR367
CARG439

site_idAC3
Number of Residues5
Detailsbinding site for residue SO4 C 503
ChainResidue
AHOH320
CSER453
CGLU454
CHOH688
CHOH806

site_idAC4
Number of Residues13
Detailsbinding site for residue 7YP C 504
ChainResidue
CHIS253
CTHR298
CTHR299
CASP398
CSER399
CSER404
CSER423
CTRP424
CGLY425
CGLY427
CGLY435
CHOH617
CHOH749

Functional Information from PROSITE/UniProt
site_idPS00134
Number of Residues6
DetailsTRYPSIN_HIS Serine proteases, trypsin family, histidine active site. VSAAHC
ChainResidueDetails
CVAL249-CYS254

site_idPS00135
Number of Residues12
DetailsTRYPSIN_SER Serine proteases, trypsin family, serine active site. DSckGDSGGPHA
ChainResidueDetails
CASP398-ALA409

site_idPS01186
Number of Residues16
DetailsEGF_2 EGF-like domain signature 2. CrCheGYslladgvsC
ChainResidueDetails
ACYS172-CYS187

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues2
DetailsGlycosylation: {"description":"N-linked (GlcNAc...) asparagine","evidences":[{"source":"PubMed","id":"19167329","evidenceCode":"ECO:0000269"},{"source":"PubMed","id":"3264725","evidenceCode":"ECO:0000269"}]}
ChainResidueDetails

site_idSWS_FT_FI2
Number of Residues3
DetailsActive site: {"description":"Charge relay system","evidences":[{"evidenceCode":"ECO:0000250"}]}
ChainResidueDetails

site_idSWS_FT_FI3
Number of Residues1
DetailsBinding site: {"evidences":[{"evidenceCode":"ECO:0000250"}]}
ChainResidueDetails

250059

PDB entries from 2026-03-04

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