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5OVI

Ras guanine nucleotide exchange factor SOS1 (Rem-cdc25) in complex with small molecule inhibitor BAY-293 (compound 23)

Functional Information from GO Data
ChainGOidnamespacecontents
A0005085molecular_functionguanyl-nucleotide exchange factor activity
A0007264biological_processsmall GTPase-mediated signal transduction
Functional Information from PDB Data
site_idAC1
Number of Residues10
Detailsbinding site for residue AXH A 2001
ChainResidue
AASN879
AHOH2296
AVAL883
ATYR884
ALEU886
AASP887
APHE890
AGLU902
AHIS905
AEDO2004

site_idAC2
Number of Residues3
Detailsbinding site for residue EDO A 2002
ChainResidue
AASP775
ATYR1031
AHOH2140

site_idAC3
Number of Residues3
Detailsbinding site for residue EDO A 2003
ChainResidue
AARG786
AGLU864
APRO1042

site_idAC4
Number of Residues5
Detailsbinding site for residue EDO A 2004
ChainResidue
ATYR884
AARG950
AAXH2001
AHOH2139
AHOH2184

Functional Information from PROSITE/UniProt
site_idPS00720
Number of Residues34
DetailsRASGEF Ras Guanine-nucleotide exchange factors domain signature. VPFfGiyLtNIlkteegnpevlkrhgkel.................INFsK
ChainResidueDetails
AVAL927-LYS960

218853

PDB entries from 2024-04-24

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