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5OVH

Ras guanine nucleotide exchange factor SOS1 (Rem-cdc25) in complex with small molecule inhibitor compound 21

Functional Information from GO Data
ChainGOidnamespacecontents
A0005085molecular_functionguanyl-nucleotide exchange factor activity
A0007264biological_processsmall GTPase-mediated signal transduction
Functional Information from PDB Data
site_idAC1
Number of Residues11
Detailsbinding site for residue AWW A 1101
ChainResidue
AMET878
AHOH1307
AHOH1338
AASN879
AVAL883
ATYR884
ALEU886
APHE890
ALEU901
AHIS905
AARG950

site_idAC2
Number of Residues3
Detailsbinding site for residue EDO A 1102
ChainResidue
AGLU903
AGLU906
ALEU907

site_idAC3
Number of Residues4
Detailsbinding site for residue EDO A 1103
ChainResidue
AASP775
ATYR1031
AHOH1233
AHOH1241

Functional Information from PROSITE/UniProt
site_idPS00720
Number of Residues34
DetailsRASGEF Ras Guanine-nucleotide exchange factors domain signature. VPFfGiyLtNIlkteegnpevlkrhgkel.................INFsK
ChainResidueDetails
AVAL927-LYS960

222415

PDB entries from 2024-07-10

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