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5OVG

Ras guanine nucleotide exchange factor SOS1 (Rem-cdc25) in complex with small molecule inhibitor compound 18

Functional Information from GO Data
ChainGOidnamespacecontents
A0005085molecular_functionguanyl-nucleotide exchange factor activity
A0007264biological_processsmall GTPase-mediated signal transduction
Functional Information from PDB Data
site_idAC1
Number of Residues7
Detailsbinding site for residue AWZ A 1101
ChainResidue
AASN879
ATYR884
AASP887
APHE890
ALEU901
AGLU902
AHIS905

site_idAC2
Number of Residues3
Detailsbinding site for residue EDO A 1102
ChainResidue
APRO1042
AARG786
AGLU864

site_idAC3
Number of Residues3
Detailsbinding site for residue EDO A 1103
ChainResidue
AASP775
ATYR1031
AHOH1206

Functional Information from PROSITE/UniProt
site_idPS00720
Number of Residues34
DetailsRASGEF Ras Guanine-nucleotide exchange factors domain signature. VPFfGiyLtNIlkteegnpevlkrhgkel.................INFsK
ChainResidueDetails
AVAL927-LYS960

218853

PDB entries from 2024-04-24

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