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5OI8

Dissociation of biochemical and antiretroviral activities of Integrase-LEDGF Allosteric Inhibitors revealed by resistance of A125 polymorphic HIV-1

Functional Information from GO Data
ChainGOidnamespacecontents
A0003676molecular_functionnucleic acid binding
A0015074biological_processDNA integration
Functional Information from PDB Data
site_idAC1
Number of Residues5
Detailsbinding site for residue MG A 301
ChainResidue
AASP64
ACAS65
AASN120
AHOH415
AHOH422

site_idAC2
Number of Residues9
Detailsbinding site for residue 9VN A 302
ChainResidue
AALA169
AGLU170
AHIS171
ATHR174
AHOH425
AGLN95
ALEU102
AALA128
AALA129

site_idAC3
Number of Residues5
Detailsbinding site for residue SO4 A 303
ChainResidue
ALYS71
AHIS171
ALEU172
AHOH402
AHOH406

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues2
DetailsBINDING: BINDING => ECO:0000250
ChainResidueDetails
AASP64
AASP116

site_idSWS_FT_FI2
Number of Residues1
DetailsBINDING: BINDING => ECO:0000250|UniProtKB:P04585
ChainResidueDetails
AGLU152

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PDB entries from 2024-07-17

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