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5OI2

Dissociation of biochemical and antiretroviral activities of Integrase-LEDGF Allosteric Inhibitors revealed by resistance of A125 polymorphic HIV-1

Functional Information from GO Data
ChainGOidnamespacecontents
A0003676molecular_functionnucleic acid binding
A0015074biological_processDNA integration
Functional Information from PDB Data
site_idAC1
Number of Residues3
Detailsbinding site for residue MG A 301
ChainResidue
AASP64
ACAS65
AASN120

site_idAC2
Number of Residues5
Detailsbinding site for residue MG A 302
ChainResidue
APRO58
AGLY59
ATRP61
APRO109
AILE204

site_idAC3
Number of Residues8
Detailsbinding site for residue MG A 303
ChainResidue
AILE84
AGLU85
AGLY106
AARG107
AVAL180
AASN184
AHOH434
ATYR83

site_idAC4
Number of Residues6
Detailsbinding site for residue MG A 304
ChainResidue
AVAL88
ATYR99
ALYS173
AVAL176
AGLN177
AHOH407

site_idAC5
Number of Residues10
Detailsbinding site for residue 9VN A 305
ChainResidue
AGLN95
ATHR124
AALA128
ATRP132
AALA169
AGLU170
AHIS171
ATHR174
AHOH426
AHOH427

site_idAC6
Number of Residues3
Detailsbinding site for residue SO4 A 306
ChainResidue
ATHR66
AHIS67
ALYS159

site_idAC7
Number of Residues6
Detailsbinding site for residue SO4 A 307
ChainResidue
ALYS71
AHIS171
ALEU172
AHOH405
AHOH411
AHOH439

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues2
DetailsBINDING: BINDING => ECO:0000250
ChainResidueDetails
AASP64
AASP116

site_idSWS_FT_FI2
Number of Residues1
DetailsBINDING: BINDING => ECO:0000250|UniProtKB:P04585
ChainResidueDetails
AGLU152

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PDB entries from 2024-07-17

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