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5O5A

Crystal structure of the human BRPF1 bromodomain in complex with BZ032

Functional Information from PDB Data
site_idAC1
Number of Residues6
Detailsbinding site for residue NO3 A 801
ChainResidue
ASER702
ALEU705
ALYS706
ATYR715
AARG722
AHOH973

site_idAC2
Number of Residues11
Detailsbinding site for residue 9LN A 802
ChainResidue
APRO656
APRO658
AGLU661
ACYS704
AASN708
APHE714
ALYS738
AHOH911
AILE652
APHE653
AGLU655

Functional Information from PROSITE/UniProt
site_idPS00633
Number of Residues58
DetailsBROMODOMAIN_1 Bromodomain signature. GniFsepvPlsevp..DYLdhIkkpMdfftMkqnleayr..Ylnfddfeedfnl.IvsNClkY
ChainResidueDetails
AGLY650-TYR707

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues104
DetailsDomain: {"description":"Bromo","evidences":[{"source":"PROSITE-ProRule","id":"PRU00035","evidenceCode":"ECO:0000255"}]}
ChainResidueDetails

243083

PDB entries from 2025-10-15

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