5O5A
Crystal structure of the human BRPF1 bromodomain in complex with BZ032
Functional Information from PDB Data
site_id | AC1 |
Number of Residues | 6 |
Details | binding site for residue NO3 A 801 |
Chain | Residue |
A | SER702 |
A | LEU705 |
A | LYS706 |
A | TYR715 |
A | ARG722 |
A | HOH973 |
site_id | AC2 |
Number of Residues | 11 |
Details | binding site for residue 9LN A 802 |
Chain | Residue |
A | PRO656 |
A | PRO658 |
A | GLU661 |
A | CYS704 |
A | ASN708 |
A | PHE714 |
A | LYS738 |
A | HOH911 |
A | ILE652 |
A | PHE653 |
A | GLU655 |
Functional Information from PROSITE/UniProt
site_id | PS00633 |
Number of Residues | 58 |
Details | BROMODOMAIN_1 Bromodomain signature. GniFsepvPlsevp..DYLdhIkkpMdfftMkqnleayr..Ylnfddfeedfnl.IvsNClkY |
Chain | Residue | Details |
A | GLY650-TYR707 |