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5O4T

Crystal structure of the human BRPF1 bromodomain in complex with BZ061

Functional Information from PDB Data
site_idAC1
Number of Residues8
Detailsbinding site for residue 9KT A 801
ChainResidue
AILE652
AVAL662
ATYR665
ACYS704
ATYR707
AASN708
APHE714
AHOH913

Functional Information from PROSITE/UniProt
site_idPS00633
Number of Residues58
DetailsBROMODOMAIN_1 Bromodomain signature. GniFsepvPlsevp..DYLdhIkkpMdfftMkqnleayr..Ylnfddfeedfnl.IvsNClkY
ChainResidueDetails
AGLY650-TYR707

237423

PDB entries from 2025-06-11

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