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5NV2

Human DNMT3B PWWP domain in complex with N-isopropyl-1,5-dimethylhexylamine (Metron S)

Functional Information from PDB Data
site_idAC1
Number of Residues4
Detailsbinding site for residue 9AE A 401
ChainResidue
AILE233
ATRP239
AASP266
AHOH508

site_idAC2
Number of Residues3
Detailsbinding site for residue SO4 A 402
ChainResidue
ALYS308
AARG312
AASN351

site_idAC3
Number of Residues2
Detailsbinding site for residue SO4 A 403
ChainResidue
AARG310
BLYS234

site_idAC4
Number of Residues5
Detailsbinding site for residue SO4 A 404
ChainResidue
ALYS251
AARG252
AHOH524
AHOH529
BHIS304

site_idAC5
Number of Residues3
Detailsbinding site for residue SO4 A 405
ChainResidue
ALYS232
ALYS234
AGLY235

site_idAC6
Number of Residues3
Detailsbinding site for residue SO4 A 406
ChainResidue
ALYS251
AARG252
BGLY265

site_idAC7
Number of Residues6
Detailsbinding site for residue 9AE B 401
ChainResidue
BILE233
BPHE236
BTRP239
BTRP263
BASP266
BSER297

site_idAC8
Number of Residues4
Detailsbinding site for residue SO4 B 402
ChainResidue
AASP275
BLYS308
BARG312
BASN351

site_idAC9
Number of Residues3
Detailsbinding site for residue SO4 B 403
ChainResidue
BLYS251
BARG252
BHOH502

site_idAD1
Number of Residues4
Detailsbinding site for residue SO4 B 404
ChainResidue
BLYS232
BLYS232
BTRP238
BTRP238

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues2
DetailsMOD_RES: Phosphoserine => ECO:0007744|PubMed:21406692, ECO:0007744|PubMed:23186163
ChainResidueDetails
ASER209
BSER209

222624

PDB entries from 2024-07-17

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