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5MQE

Crystal structure of CREBBP bromodomain complexed with CBP006

Functional Information from GO Data
ChainGOidnamespacecontents
A0004402molecular_functionhistone acetyltransferase activity
A0006355biological_processregulation of DNA-templated transcription
B0004402molecular_functionhistone acetyltransferase activity
B0006355biological_processregulation of DNA-templated transcription
Functional Information from PDB Data
site_idAC1
Number of Residues5
Detailsbinding site for residue PKU A 1201
ChainResidue
AVAL1115
AASN1168
AVAL1174
AHOH1317
AHOH1343

site_idAC2
Number of Residues5
Detailsbinding site for residue PKU B 1201
ChainResidue
BHOH1343
BPRO1110
BASN1168
BVAL1174
BHOH1311

Functional Information from PROSITE/UniProt
site_idPS00633
Number of Residues60
DetailsBROMODOMAIN_1 Bromodomain signature. SlpFrqpvDpqllgipDYFdiVknpMdlstIkrkldtgq..Yqepwqyvddvwl.MfnNAwlY
ChainResidueDetails
ASER1108-TYR1167

237735

PDB entries from 2025-06-18

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