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5MNN

Cationic trypsin in complex with N-amidinopiperidine (deuterated sample at 100 K)

Functional Information from GO Data
ChainGOidnamespacecontents
A0004175molecular_functionendopeptidase activity
A0004252molecular_functionserine-type endopeptidase activity
A0005515molecular_functionprotein binding
A0005576cellular_componentextracellular region
A0005615cellular_componentextracellular space
A0006508biological_processproteolysis
A0007586biological_processdigestion
A0008236molecular_functionserine-type peptidase activity
A0046872molecular_functionmetal ion binding
A0097180cellular_componentserine protease inhibitor complex
A0097655molecular_functionserpin family protein binding
Functional Information from PDB Data
site_idAC1
Number of Residues6
Detailsbinding site for residue CA A 301
ChainResidue
AGLU70
AASN72
AVAL75
AGLU80
AHOH411
AHOH535

site_idAC2
Number of Residues15
Detailsbinding site for residue MRZ A 302
ChainResidue
AGLN192
ASER195
AVAL213
ATRP215
AGLY216
AGLY219
ACYS220
AGLY226
ASO4305
AHOH444
AHOH551
AHOH645
AASP189
ASER190
ACYS191

site_idAC3
Number of Residues7
Detailsbinding site for residue SO4 A 303
ChainResidue
ALYS87
ALYS107
ATHR149
ATYR151
AHOH403
AHOH410
AHOH441

site_idAC4
Number of Residues8
Detailsbinding site for residue SO4 A 304
ChainResidue
ALYS169
APRO173
AGLY174
AHOH473
AHOH479
AHOH513
AHOH544
AHOH641

site_idAC5
Number of Residues5
Detailsbinding site for residue SO4 A 305
ChainResidue
AHIS57
AGLN192
AGLY193
ASER195
AMRZ302

site_idAC6
Number of Residues10
Detailsbinding site for residue SO4 A 306
ChainResidue
APRO124
ATHR125
ASER127
ASER147
AGLY148
ALYS204
AHOH486
AHOH523
AHOH524
AHOH533

Functional Information from PROSITE/UniProt
site_idPS00134
Number of Residues6
DetailsTRYPSIN_HIS Serine proteases, trypsin family, histidine active site. VSAAHC
ChainResidueDetails
AVAL53-CYS58

site_idPS00135
Number of Residues12
DetailsTRYPSIN_SER Serine proteases, trypsin family, serine active site. DScqGDSGGPVV
ChainResidueDetails
AASP189-VAL200

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues3
DetailsACT_SITE: Charge relay system
ChainResidueDetails
AHIS57
AASP102
ASER195

site_idSWS_FT_FI2
Number of Residues7
DetailsBINDING:
ChainResidueDetails
AGLU70
AASN72
AVAL75
AGLU80
AASP189
AGLN192
ASER195

224572

PDB entries from 2024-09-04

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