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5MMO

E. coli DNA Gyrase B 24 kDa ATPase domain in complex with [3-(3-ethyl-ureido)-5-(pyridin-4-yl)-isoquinolin-8-yl-methyl]-carbamic acid prop-2-ynyl ester

Functional Information from GO Data
ChainGOidnamespacecontents
A0003677molecular_functionDNA binding
A0003918molecular_functionDNA topoisomerase type II (double strand cut, ATP-hydrolyzing) activity
A0005524molecular_functionATP binding
A0006265biological_processDNA topological change
Functional Information from PDB Data
site_idAC1
Number of Residues15
Detailsbinding site for residue 9JG A 301
ChainResidue
AASN46
AARG136
ATHR165
APO4302
AHOH417
AHOH462
AHOH472
AGLU50
AVAL71
AASP73
AARG76
AGLY77
AILE78
APRO79
AILE94

site_idAC2
Number of Residues6
Detailsbinding site for residue PO4 A 302
ChainResidue
APRO79
ATHR80
AGLY81
AARG136
AGLU137
A9JG301

Catalytic Information from CSA
site_idMCSA1
Number of Residues
DetailsM-CSA 745
ChainResidueDetails

224004

PDB entries from 2024-08-21

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