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5M6N

Small Molecule inhibitors of IAP

Functional Information from PDB Data
site_idAC1
Number of Residues4
Detailsbinding site for residue ZN A 1001
ChainResidue
ACYS300
ACYS303
AHIS320
ACYS327

site_idAC2
Number of Residues5
Detailsbinding site for residue SO4 A 1002
ChainResidue
AHIS259
AMET260
AHOH1113
AHOH1123
AHOH1203

site_idAC3
Number of Residues9
Detailsbinding site for residue SO4 A 1003
ChainResidue
AHIS348
AGLU351
AHOH1129
AHOH1133
AHOH1143
BGLU282
BGLN283
BSER286
BHOH1126

site_idAC4
Number of Residues18
Detailsbinding site for residue 7H9 A 1004
ChainResidue
AGLN261
AASP297
AVAL298
ALYS299
AGLY306
ALEU307
AARG308
ACYS309
ATRP310
AASP314
AGLU319
ATRP323
APHE324
AHOH1179
AHOH1217
AHOH1248
BARG268
BMET271

site_idAC5
Number of Residues4
Detailsbinding site for residue ZN B 1001
ChainResidue
BCYS300
BCYS303
BHIS320
BCYS327

site_idAC6
Number of Residues4
Detailsbinding site for residue SO4 B 1002
ChainResidue
BTHR262
BALA265
BARG268
BHOH1128

site_idAC7
Number of Residues5
Detailsbinding site for residue SO4 B 1003
ChainResidue
BTHR262
BHIS263
BHOH1103
BHOH1120
BHOH1134

site_idAC8
Number of Residues7
Detailsbinding site for residue SO4 B 1004
ChainResidue
ALYS322
ATRP323
AARG332
BMET271
BTYR272
BHOH1117
BHOH1169

site_idAC9
Number of Residues18
Detailsbinding site for residue 7H9 B 1005
ChainResidue
ALEU350
AHOH1287
BASP297
BVAL298
BLYS299
BGLY306
BLEU307
BARG308
BCYS309
BTRP310
BASP314
BGLU319
BTRP323
BPHE324
BHOH1107
BHOH1139
BHOH1144
BHOH1173

Functional Information from PROSITE/UniProt
site_idPS01282
Number of Residues68
DetailsBIR_REPEAT_1 BIR repeat. HaaRmrtfmy.Wpssvpvqpeqlas.AGFyYvgrnDdvkCfcCdgglrcWesgddpwveHakwfPrCefL
ChainResidueDetails
AHIS263-LEU330

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues8
DetailsBINDING:
ChainResidueDetails
ACYS300
ACYS303
AHIS320
ACYS327
BCYS300
BCYS303
BHIS320
BCYS327

223532

PDB entries from 2024-08-07

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