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5M6H

Small Molecule inhibitors of IAP

Functional Information from PDB Data
site_idAC1
Number of Residues4
Detailsbinding site for residue ZN A 401
ChainResidue
ACYS300
ACYS303
AHIS320
ACYS327

site_idAC2
Number of Residues6
Detailsbinding site for residue NA A 402
ChainResidue
AHOH555
APHE272
APHE272
AHOH538
AHOH538
AHOH555

site_idAC3
Number of Residues12
Detailsbinding site for residue 7J6 A 403
ChainResidue
ALEU292
AVAL298
AGLY306
ALEU307
ATHR308
AASP309
ATRP310
ALYS311
AGLU314
AGLN319
ATRP323
ATYR324

Functional Information from PROSITE/UniProt
site_idPS01282
Number of Residues66
DetailsBIR_REPEAT_1 BIR repeat. YeaRiftfgt.Wiysvnkeqlar...AGFyAlgegDkvkCfhCgggltdWkpsedpweqHakwyPgCkyL
ChainResidueDetails
ATYR265-LEU330

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues65
DetailsRepeat: {"description":"BIR 3"}
ChainResidueDetails

site_idSWS_FT_FI2
Number of Residues15
DetailsRegion: {"description":"Required for interaction with SEPTIN4 isoform ARTS","evidences":[{"source":"PubMed","id":"21695558","evidenceCode":"ECO:0000269"}]}
ChainResidueDetails

site_idSWS_FT_FI3
Number of Residues21
DetailsRegion: {"description":"Required for interaction with DIABLO","evidences":[{"source":"PubMed","id":"21695558","evidenceCode":"ECO:0000269"}]}
ChainResidueDetails

site_idSWS_FT_FI4
Number of Residues4
DetailsBinding site: {"evidences":[{"source":"PROSITE-ProRule","id":"PRU00029","evidenceCode":"ECO:0000255"}]}
ChainResidueDetails

site_idSWS_FT_FI5
Number of Residues3
DetailsCross-link: {"description":"Glycyl lysine isopeptide (Lys-Gly) (interchain with G-Cter in ubiquitin)","evidences":[{"source":"PubMed","id":"12747801","evidenceCode":"ECO:0000269"}]}
ChainResidueDetails

239803

PDB entries from 2025-08-06

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