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5M6E

Small Molecule inhibitors of IAP

Functional Information from PDB Data
site_idAC1
Number of Residues4
Detailsbinding site for residue ZN A 401
ChainResidue
ACYS300
ACYS303
AHIS320
ACYS327

site_idAC2
Number of Residues4
Detailsbinding site for residue NA A 402
ChainResidue
APHE272
APHE272
AHOH610
AHOH610

site_idAC3
Number of Residues3
Detailsbinding site for residue DMS A 403
ChainResidue
AGLY306
A7HT404
AMET248

site_idAC4
Number of Residues14
Detailsbinding site for residue 7HT A 404
ChainResidue
ALEU292
AGLY306
ALEU307
ATHR308
AASP309
ATRP310
AGLU314
AGLN319
ATRP323
ATYR324
ADMS403
AHOH506
AHOH517
AHOH570

Functional Information from PROSITE/UniProt
site_idPS01282
Number of Residues66
DetailsBIR_REPEAT_1 BIR repeat. YeaRiftfgt.Wiysvnkeqlar...AGFyAlgegDkvkCfhCgggltdWkpsedpweqHakwyPgCkyL
ChainResidueDetails
ATYR265-LEU330

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues4
DetailsBINDING: BINDING => ECO:0000255|PROSITE-ProRule:PRU00029
ChainResidueDetails
ACYS300
ACYS303
AHIS320
ACYS327

site_idSWS_FT_FI2
Number of Residues3
DetailsCROSSLNK: Glycyl lysine isopeptide (Lys-Gly) (interchain with G-Cter in ubiquitin) => ECO:0000269|PubMed:12747801
ChainResidueDetails
ALYS322
ALYS328

223532

PDB entries from 2024-08-07

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