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5LJ2

N-TERMINAL BROMODOMAIN OF HUMAN BRD4 WITH 5-(5-aminopyridin-3-yl)-8-(((3R,4R)-3-((1,1-dioxidotetrahydro-2H-thiopyran-4-yl)methoxy)piperidin-4-yl)amino)-3-methyl-1,7-naphthyridin-2(1H)-one

Functional Information from PDB Data
site_idAC1
Number of Residues6
Detailsbinding site for residue EDO A 201
ChainResidue
AGLN123
AILE126
AHOH304
AHOH316
AHOH333
AHOH465

site_idAC2
Number of Residues7
Detailsbinding site for residue EDO A 202
ChainResidue
ATHR103
AASN135
AHOH314
AHOH319
AILE100
AILE101
ALYS102

site_idAC3
Number of Residues4
Detailsbinding site for residue EDO A 203
ChainResidue
AILE138
AGLN159
ALYS160
AHOH311

site_idAC4
Number of Residues16
Detailsbinding site for residue 6XW A 204
ChainResidue
ALYS57
AARG58
AGLN59
ATRP81
AGLN85
ALEU92
ALYS99
AASN140
AASP144
AILE146
AHOH302
AHOH344
AHOH349
AHOH359
AHOH419
AHOH424

Functional Information from PROSITE/UniProt
site_idPS00633
Number of Residues60
DetailsBROMODOMAIN_1 Bromodomain signature. AwpFqqpvDavklnlpDYYkiIktpMdmgtIkkrlenny..Ywnaqeciqdfnt.MftNCyiY
ChainResidueDetails
AALA80-TYR139

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues106
DetailsDomain: {"description":"Bromo 1","evidences":[{"source":"PROSITE-ProRule","id":"PRU00035","evidenceCode":"ECO:0000255"}]}
ChainResidueDetails

site_idSWS_FT_FI2
Number of Residues1
DetailsSite: {"description":"Acetylated histone binding","evidences":[{"source":"PubMed","id":"22464331","evidenceCode":"ECO:0000269"}]}
ChainResidueDetails

site_idSWS_FT_FI3
Number of Residues2
DetailsCross-link: {"description":"Glycyl lysine isopeptide (Lys-Gly) (interchain with G-Cter in SUMO2)","evidences":[{"source":"PubMed","id":"28112733","evidenceCode":"ECO:0007744"}]}
ChainResidueDetails

243083

PDB entries from 2025-10-15

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