Loading
PDBj
MenuPDBj@FacebookPDBj@X(formerly Twitter)PDBj@BlueSkyPDBj@YouTubewwPDB FoundationwwPDBDonate
RCSB PDBPDBeBMRBAdv. SearchSearch help

5LAZ

Novel Spiro[3H-indole-3,2 -pyrrolidin]-2(1H)-one Inhibitors of the MDM2-p53 Interaction: HDM2 (MDM2) IN COMPLEX WITH COMPOUND BI-0252

Functional Information from GO Data
ChainGOidnamespacecontents
A0005634cellular_componentnucleus
A0043066biological_processnegative regulation of apoptotic process
A0051726biological_processregulation of cell cycle
Functional Information from PDB Data
site_idAC1
Number of Residues11
Detailsbinding site for residue 6ST A 201
ChainResidue
ALEU54
ATYR100
AHOH327
AILE61
AMET62
APHE86
AVAL93
ALYS94
ALYS94
AHIS96
AILE99

site_idAC2
Number of Residues5
Detailsbinding site for residue ZN A 202
ChainResidue
AHIS73
AHIS73
ALYS94
AHOH303
AHOH303

site_idAC3
Number of Residues7
Detailsbinding site for residue SO4 A 203
ChainResidue
APRO20
AALA21
ALYS51
ALYS51
AHOH305
AHOH305
AHOH312

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues83
DetailsDomain: {"description":"SWIB/MDM2","evidences":[{"source":"PROSITE-ProRule","id":"PRU01273","evidenceCode":"ECO:0000255"}]}
ChainResidueDetails

248335

PDB entries from 2026-01-28

PDB statisticsPDBj update infoContact PDBjnumon