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5KRT

HIV-1 Integrase Catalytic Core Domain (CCD) in Complex with a Fragment-Derived Allosteric Inhibitor

Functional Information from GO Data
ChainGOidnamespacecontents
A0003676molecular_functionnucleic acid binding
A0015074biological_processDNA integration
Functional Information from PDB Data
site_idAC1
Number of Residues7
Detailsbinding site for residue 6W6 A 301
ChainResidue
ATHR122
ASER123
ATHR124
AGLU157
AGLN164
AILE182
ALYS186

site_idAC2
Number of Residues10
Detailsbinding site for residue 6W6 A 302
ChainResidue
ATYR99
ALEU102
ATHR125
AALA128
AALA169
AGLU170
AHIS171
ATHR174
AGLN95
AALA98

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues2
DetailsBINDING:
ChainResidueDetails
AASP64
AASP116

site_idSWS_FT_FI2
Number of Residues1
DetailsBINDING: BINDING => ECO:0000250|UniProtKB:P04585
ChainResidueDetails
AGLU152

221716

PDB entries from 2024-06-26

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