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5KGW

HIV1 catalytic core domain in complex with inhibitor: (2~{S})-2-[3-(3,4-dihydro-2~{H}-chromen-6-yl)-1-methyl-indol-2-yl]-2-[(2-methylpropan-2-yl)oxy]ethanoic acid

Functional Information from GO Data
ChainGOidnamespacecontents
A0003676molecular_functionnucleic acid binding
A0015074biological_processDNA integration
Functional Information from PDB Data
site_idAC1
Number of Residues5
Detailsbinding site for residue SO4 A 301
ChainResidue
ALYS71
AARG166
AHIS171
ALEU172
AHOH409

site_idAC2
Number of Residues2
Detailsbinding site for residue SO4 A 302
ChainResidue
ATHR66
AHIS67

site_idAC3
Number of Residues6
Detailsbinding site for residue SO4 A 303
ChainResidue
ASER123
ATHR125
ALYS186
AHOH422
ATHR93
AGLY94

site_idAC4
Number of Residues10
Detailsbinding site for residue 7SK A 304
ChainResidue
AGLN95
ALEU102
ATHR125
AALA129
ATRP132
AALA169
AGLU170
AHIS171
ATHR174
AMET178

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues2
DetailsBinding site: {}
ChainResidueDetails

site_idSWS_FT_FI2
Number of Residues1
DetailsBinding site: {"evidences":[{"source":"UniProtKB","id":"P04585","evidenceCode":"ECO:0000250"}]}
ChainResidueDetails

247536

PDB entries from 2026-01-14

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