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5ISL

Linked KDM5A Jmj Domain Bound to the Inhibitor C49 (2-{[(2-{[(E)-2-(dimethylamino)ethenyl](ethyl)amino}-2-oxoethyl)amino]methyl}pyridine-4-carboxylic acid)

Functional Information from PDB Data
site_idAC1
Number of Residues16
Detailsbinding site for residue MMK A 601
ChainResidue
ATYR409
AVAL584
AASN585
AMN602
AHOH731
AHOH734
AHOH778
AHOH822
ATRP470
ATYR472
APHE480
AHIS483
AGLU485
ALYS501
ATRP503
AHIS571

site_idAC2
Number of Residues5
Detailsbinding site for residue MN A 602
ChainResidue
AHIS483
AGLU485
AHIS571
AMMK601
AHOH731

site_idAC3
Number of Residues9
Detailsbinding site for residue GOL A 603
ChainResidue
ASER375
AMET380
APRO381
AGLU485
AHIS487
ATRP488
AHOH703
AHOH708
AHOH727

site_idAC4
Number of Residues5
Detailsbinding site for residue EDO A 604
ChainResidue
ASER399
AILE539
AMET540
AASN541
AHOH772

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues41
DetailsDomain: {"description":"JmjN","evidences":[{"source":"PROSITE-ProRule","id":"PRU00537","evidenceCode":"ECO:0000255"}]}
ChainResidueDetails

site_idSWS_FT_FI2
Number of Residues4
DetailsMotif: {"description":"GSGFP motif","evidences":[{"source":"UniProtKB","id":"Q3UXZ9","evidenceCode":"ECO:0000250"}]}
ChainResidueDetails

site_idSWS_FT_FI3
Number of Residues4
DetailsBinding site: {"evidences":[{"source":"PubMed","id":"26645689","evidenceCode":"ECO:0000269"},{"source":"PubMed","id":"27427228","evidenceCode":"ECO:0000269"}]}
ChainResidueDetails

site_idSWS_FT_FI4
Number of Residues2
DetailsBinding site: {"evidences":[{"source":"PROSITE-ProRule","id":"PRU00538","evidenceCode":"ECO:0000255"},{"source":"PubMed","id":"26645689","evidenceCode":"ECO:0000305"},{"source":"PubMed","id":"27214401","evidenceCode":"ECO:0000305"},{"source":"PubMed","id":"27427228","evidenceCode":"ECO:0000305"},{"source":"PubMed","id":"27499454","evidenceCode":"ECO:0000305"}]}
ChainResidueDetails

site_idSWS_FT_FI5
Number of Residues1
DetailsBinding site: {"evidences":[{"source":"PubMed","id":"26645689","evidenceCode":"ECO:0000305"},{"source":"PubMed","id":"27214401","evidenceCode":"ECO:0000305"},{"source":"PubMed","id":"27427228","evidenceCode":"ECO:0000305"},{"source":"PubMed","id":"27499454","evidenceCode":"ECO:0000305"}]}
ChainResidueDetails

243083

PDB entries from 2025-10-15

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