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5IH0

Macrolide 2'-phosphotransferase type II Y92M mutant - complex with GDP and erythromycin

Functional Information from GO Data
ChainGOidnamespacecontents
A0016740molecular_functiontransferase activity
A0046872molecular_functionmetal ion binding
Functional Information from PDB Data
site_idAC1
Number of Residues5
Detailsbinding site for residue MG A 401
ChainResidue
AHIS205
AASP219
AGDP403
AHOH645
AHOH705

site_idAC2
Number of Residues5
Detailsbinding site for residue ACT A 402
ChainResidue
AHOH562
APHE33
AARG49
AARG59
AHOH534

site_idAC3
Number of Residues18
Detailsbinding site for residue GDP A 403
ChainResidue
APHE33
APHE37
AARG49
ALYS94
ALEU95
AHIS205
AASP219
AMG401
AHOH506
AHOH524
AHOH556
AHOH560
AHOH604
AHOH615
AHOH645
AHOH705
AHOH714
AHOH725

site_idAC4
Number of Residues20
Detailsbinding site for residue ERY A 404
ChainResidue
AHIS105
AGLY108
AASN109
ATYR110
AASP200
AVAL201
AHIS202
AGLU222
AHIS230
AILE233
AARG237
ATYR273
ASER276
AILE277
AMET292
AHOH573
AHOH581
AHOH609
AHOH633
AHOH661

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PDB entries from 2024-07-24

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