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5HRW

Crystal structure of the fifth bromodomain of human PB1 in complex with 1-propylisochromeno[3,4-c]pyrazol-5(2H)-one) compound

Functional Information from GO Data
ChainGOidnamespacecontents
A0006338biological_processchromatin remodeling
A0016586cellular_componentRSC-type complex
B0006338biological_processchromatin remodeling
B0016586cellular_componentRSC-type complex
Functional Information from PDB Data
site_idAC1
Number of Residues14
Detailsbinding site for residue 64E A 801
ChainResidue
AILE683
AASN739
AILE745
AHOH911
AHOH923
BEDO802
APHE684
ALEU687
ATYR696
AMET704
AASP705
AMET731
AALA735
ATYR738

site_idAC2
Number of Residues2
Detailsbinding site for residue EDO A 802
ChainResidue
AARG686
AEDO803

site_idAC3
Number of Residues3
Detailsbinding site for residue EDO A 803
ChainResidue
AARG686
AEDO802
BARG676

site_idAC4
Number of Residues4
Detailsbinding site for residue EDO A 804
ChainResidue
ALEU693
APRO694
AASP695
ATYR738

site_idAC5
Number of Residues3
Detailsbinding site for residue EDO A 805
ChainResidue
AMET655
AASN663
AGLU664

site_idAC6
Number of Residues6
Detailsbinding site for residue SO4 A 806
ChainResidue
APHE732
AASN733
ACYS736
AALA749
ALEU750
AHIS753

site_idAC7
Number of Residues12
Detailsbinding site for residue 64E B 801
ChainResidue
BILE683
BPHE684
BLEU687
BTYR696
BMET704
BMET731
BALA735
BTYR738
BASN739
BILE745
BHOH904
BHOH916

site_idAC8
Number of Residues5
Detailsbinding site for residue EDO B 802
ChainResidue
A64E801
AHOH918
BSER743
BLEU744
BHOH906

Functional Information from PROSITE/UniProt
site_idPS00633
Number of Residues58
DetailsBROMODOMAIN_1 Bromodomain signature. SaiFlrlpSrselp..DYYltIkkpMdmekIrshmmank..Yqdidsmvedfvm.MfnNActY
ChainResidueDetails
ASER681-TYR738

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues2
DetailsModified residue: {"description":"Phosphoserine","evidences":[{"source":"PubMed","id":"23186163","evidenceCode":"ECO:0007744"}]}
ChainResidueDetails

247536

PDB entries from 2026-01-14

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