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5HRP

HIV Integrase Catalytic Domain containing F185K + A124T mutations complexed with GSK0002

Functional Information from GO Data
ChainGOidnamespacecontents
A0003676molecular_functionnucleic acid binding
A0015074biological_processDNA integration
Functional Information from PDB Data
site_idAC1
Number of Residues4
Detailsbinding site for residue CAC A 301
ChainResidue
ACYS65
AGLU92
ATHR97
AASN120

site_idAC2
Number of Residues4
Detailsbinding site for residue CAC A 302
ChainResidue
ACYS130
AILE135
ALYS136
AGLN137

site_idAC3
Number of Residues6
Detailsbinding site for residue SO4 A 303
ChainResidue
AGLU170
AHIS171
ALEU172
AHOH419
AHOH463
ALYS71

site_idAC4
Number of Residues4
Detailsbinding site for residue SO4 A 304
ChainResidue
AALA128
ATRP131
A65P310
AHOH411

site_idAC5
Number of Residues5
Detailsbinding site for residue SO4 A 305
ChainResidue
ATHR124
ALYS160
AGLN164
AEDO307
AHOH423

site_idAC6
Number of Residues2
Detailsbinding site for residue SO4 A 306
ChainResidue
ATHR66
AHIS67

site_idAC7
Number of Residues5
Detailsbinding site for residue EDO A 307
ChainResidue
ASER123
ATHR124
ATHR125
ASO4305
AHOH426

site_idAC8
Number of Residues3
Detailsbinding site for residue EDO A 308
ChainResidue
AASP167
AGLN168
AHOH411

site_idAC9
Number of Residues3
Detailsbinding site for residue EDO A 309
ChainResidue
AARG166
AALA169
AGLU170

site_idAD1
Number of Residues14
Detailsbinding site for residue 65P A 310
ChainResidue
ALEU102
ATHR124
ATHR125
AALA129
ATRP132
AGLN168
AALA169
AGLU170
AHIS171
ATHR174
ASO4304
AHOH409
AHOH442
AHOH470

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues2
DetailsBINDING: BINDING => ECO:0000250
ChainResidueDetails
AASP64
AASP116

site_idSWS_FT_FI2
Number of Residues1
DetailsBINDING: BINDING => ECO:0000305
ChainResidueDetails
AGLU152

Catalytic Information from CSA
site_idMCSA1
Number of Residues
DetailsM-CSA 175
ChainResidueDetails

219140

PDB entries from 2024-05-01

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