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5GTO

Human PPARgamma ligand binding dmain complexed with S35

Functional Information from GO Data
ChainGOidnamespacecontents
A0003677molecular_functionDNA binding
A0004879molecular_functionnuclear receptor activity
A0005634cellular_componentnucleus
A0006355biological_processregulation of DNA-templated transcription
Functional Information from PDB Data
site_idAC1
Number of Residues16
Detailsbinding site for residue T35 A 501
ChainResidue
ASER245
AILE281
AGLN283
AGLY284
ALEU340
AILE341
ASER342
AMYR502
AGLU259
AILE262
APHE264
AILE267
ATHR268
APRO269
ALEU270
AARG280

site_idAC2
Number of Residues8
Detailsbinding site for residue MYR A 502
ChainResidue
ALEU228
ACYS285
ASER289
AMET329
ALEU333
AT35501
AGOL503
AHOH610

site_idAC3
Number of Residues8
Detailsbinding site for residue GOL A 503
ChainResidue
APHE282
AGLN286
ASER289
AHIS323
AHIS449
ALEU469
ATYR473
AMYR502

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues1
DetailsMOD_RES: Phosphoserine => ECO:0007744|PubMed:23186163
ChainResidueDetails
BSER698
AHIS323
AHIS449
ATYR473

site_idSWS_FT_FI2
Number of Residues2
DetailsCROSSLNK: Glycyl lysine isopeptide (Lys-Gly) (interchain with G-Cter in ubiquitin) => ECO:0000269|PubMed:36737649
ChainResidueDetails
ALYS224

220113

PDB entries from 2024-05-22

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