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5GI9

Crystal Structure of Drosophila melanogaster Dopamine N-Acetyltransferase in Ternary Complex with CoA and Acetyl-Tryptamine

Functional Information from GO Data
ChainGOidnamespacecontents
A0016747molecular_functionacyltransferase activity, transferring groups other than amino-acyl groups
Functional Information from PDB Data
site_idAC1
Number of Residues36
Detailsbinding site for residue COA A 301
ChainResidue
AASP46
ALEU155
AGLY156
AILE157
AALA158
ACYS181
ASER182
ASER186
AVAL189
ALYS192
A7AN302
APRO48
AD1D304
AHOH421
AHOH433
AHOH435
AHOH436
AHOH445
AHOH455
AHOH456
AHOH460
AHOH466
AASP132
AHOH473
AHOH483
AHOH493
AHOH498
AHOH512
AHOH535
AHOH544
AVAL133
ALEU146
ASER147
AVAL148
AARG153
AGLY154

site_idAC2
Number of Residues13
Detailsbinding site for residue 7AN A 302
ChainResidue
APHE43
AGLU47
AASN50
ALEU61
APHE114
AILE117
AMET121
AGLY143
ALYS144
AILE145
ALEU146
ALEU180
ACOA301

site_idAC3
Number of Residues10
Detailsbinding site for residue 7AN A 303
ChainResidue
ATHR41
APHE42
AGLU197
AARG200
AMET201
AGLN202
AVAL221
AGLY222
AILE223
AGLN224

site_idAC4
Number of Residues8
Detailsbinding site for residue D1D A 304
ChainResidue
APRO48
AHIS196
AGLU229
ACOA301
AHOH446
AHOH480
AHOH495
AHOH512

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues2
DetailsBINDING: BINDING => ECO:0000269|PubMed:22716280, ECO:0007744|PDB:3TE4
ChainResidueDetails
ALEU146
AGLY154

site_idSWS_FT_FI2
Number of Residues3
DetailsSITE: Has a role in the catalytic activity => ECO:0000269|PubMed:25406072
ChainResidueDetails
AGLU47
ASER182
ASER186

site_idSWS_FT_FI3
Number of Residues1
DetailsSITE: Might be involved in substrate binding => ECO:0000269|PubMed:25406072
ChainResidueDetails
ATYR64

site_idSWS_FT_FI4
Number of Residues1
DetailsSITE: Regulates binding affinity for coenzyme A (CoASH) => ECO:0000269|PubMed:25406072
ChainResidueDetails
AARG153

site_idSWS_FT_FI5
Number of Residues1
DetailsSITE: Acetyl-CoA => ECO:0000269|PubMed:22716280, ECO:0007744|PDB:3TE4
ChainResidueDetails
ALYS192

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PDB entries from 2024-07-17

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