5G4S

BROMODOMAIN OF HUMAN BRPF1 WITH N-1,3-dimethyl-6-2R-2- methylpiperazin-1-yl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl-N- ethyl-2-methoxybenzamide

Functional Information from PDB Data

site_id	AC1
Number of Residues	1
Details	BINDING SITE FOR RESIDUE EDO A 1800

Chain	Residue
A	GLU695

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site_id	AC2
Number of Residues	14
Details	BINDING SITE FOR RESIDUE 8VI A 1739

Chain	Residue
A	PHE676
A	TYR707
A	ASN708
A	PHE714
A	HOH2057
A	HOH2125
A	ILE624
A	MET626
A	ASN651
A	ILE652
A	GLU655
A	VAL657
A	PRO658
A	VAL662

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Functional Information from PROSITE/UniProt

site_id	PS00633
Number of Residues	58
Details	BROMODOMAIN_1 Bromodomain signature. GniFsepvPlsevp..DYLdhIkkpMdfftMkqnleayr..Ylnfddfeedfnl.IvsNClkY

Chain	Residue	Details
A	GLY650-TYR707

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Functional Information from SwissProt/UniProt

site_id	SWS_FT_FI1
Number of Residues	104
Details	Domain: {"description":"Bromo","evidences":[{"source":"PROSITE-ProRule","id":"PRU00035","evidenceCode":"ECO:0000255"}]}

Chain

Residue

Details

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