5G4S
BROMODOMAIN OF HUMAN BRPF1 WITH N-1,3-dimethyl-6-2R-2- methylpiperazin-1-yl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl-N- ethyl-2-methoxybenzamide
Functional Information from PDB Data
| site_id | AC1 |
| Number of Residues | 1 |
| Details | BINDING SITE FOR RESIDUE EDO A 1800 |
| Chain | Residue |
| A | GLU695 |
| site_id | AC2 |
| Number of Residues | 14 |
| Details | BINDING SITE FOR RESIDUE 8VI A 1739 |
| Chain | Residue |
| A | PHE676 |
| A | TYR707 |
| A | ASN708 |
| A | PHE714 |
| A | HOH2057 |
| A | HOH2125 |
| A | ILE624 |
| A | MET626 |
| A | ASN651 |
| A | ILE652 |
| A | GLU655 |
| A | VAL657 |
| A | PRO658 |
| A | VAL662 |
Functional Information from PROSITE/UniProt
| site_id | PS00633 |
| Number of Residues | 58 |
| Details | BROMODOMAIN_1 Bromodomain signature. GniFsepvPlsevp..DYLdhIkkpMdfftMkqnleayr..Ylnfddfeedfnl.IvsNClkY |
| Chain | Residue | Details |
| A | GLY650-TYR707 |
