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5G0H

Crystal structure of Danio rerio HDAC6 CD2 in complex with (S)- trichostatin A

Functional Information from GO Data
ChainGOidnamespacecontents
A0000118cellular_componenthistone deacetylase complex
A0004407molecular_functionhistone deacetylase activity
A0006325biological_processchromatin organization
A0016575biological_processhistone deacetylation
Functional Information from PDB Data
site_idAC1
Number of Residues14
DetailsBINDING SITE FOR RESIDUE E1Z A 1801
ChainResidue
ASER531
AASP705
ATYR745
AZN1804
AEDO1813
AHOH2190
AHIS573
AHIS574
AGLY582
APHE583
AASP612
AHIS614
APHE643
AASN645

site_idAC2
Number of Residues5
DetailsBINDING SITE FOR RESIDUE K A 1802
ChainResidue
AASP610
AASP612
AHIS614
ASER633
ALEU634

site_idAC3
Number of Residues6
DetailsBINDING SITE FOR RESIDUE K A 1803
ChainResidue
APHE623
AASP626
AVAL629
ATYR662
AHOH2195
AHOH2199

site_idAC4
Number of Residues4
DetailsBINDING SITE FOR RESIDUE ZN A 1804
ChainResidue
AASP612
AHIS614
AASP705
AE1Z1801

site_idAC5
Number of Residues6
DetailsBINDING SITE FOR RESIDUE EDO A 1805
ChainResidue
ALEU557
ATHR600
ALEU604
AHOH2124
AHOH2125
AHOH2283

site_idAC6
Number of Residues9
DetailsBINDING SITE FOR RESIDUE EDO A 1806
ChainResidue
ASER505
ALYS506
APRO676
AMET679
AASP770
ATHR773
AHOH2077
AHOH2258
AHOH2328

site_idAC7
Number of Residues2
DetailsBINDING SITE FOR RESIDUE EDO A 1807
ChainResidue
AASN784
AASN800

site_idAC8
Number of Residues6
DetailsBINDING SITE FOR RESIDUE EDO A 1808
ChainResidue
AHIS456
AASN457
ASER461
APRO467
AHOH2015
AHOH2022

site_idAC9
Number of Residues5
DetailsBINDING SITE FOR RESIDUE EDO A 1809
ChainResidue
ALYS672
AGLY674
AGLU677
AGLN716
AHOH2295

site_idBC1
Number of Residues5
DetailsBINDING SITE FOR RESIDUE EDO A 1810
ChainResidue
AARG660
ATYR662
APHE793
ATRP794
AHOH2026

site_idBC2
Number of Residues3
DetailsBINDING SITE FOR RESIDUE EDO A 1811
ChainResidue
ATRP459
AASP460
AHIS462

site_idBC3
Number of Residues4
DetailsBINDING SITE FOR RESIDUE EDO A 1812
ChainResidue
APRO442
AMET730
ALEU761
AHOH2352

site_idBC4
Number of Residues5
DetailsBINDING SITE FOR RESIDUE EDO A 1813
ChainResidue
ATYR529
AASN530
ASER531
AE1Z1801
AHOH2103

site_idBC5
Number of Residues7
DetailsBINDING SITE FOR RESIDUE EDO A 1814
ChainResidue
ASER461
AHIS462
ALEU466
AARG660
APHE793
AHOH2025
AHOH2345

220472

PDB entries from 2024-05-29

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