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5FPE

Structure of heat shock-related 70kDA protein 2 with small-molecule ligand 1H-1,2,4-triazol-3-amine (AT485) in an alternate binding site.

Functional Information from GO Data
ChainGOidnamespacecontents
A0005524molecular_functionATP binding
A0140662molecular_functionATP-dependent protein folding chaperone
B0005524molecular_functionATP binding
B0140662molecular_functionATP-dependent protein folding chaperone
Functional Information from PDB Data
site_idAC1
Number of Residues5
DetailsBINDING SITE FOR RESIDUE 3TR B 1385
ChainResidue
BTYR149
BASP208
BALA225
BHOH2268
BHOH2269

site_idAC2
Number of Residues5
DetailsBINDING SITE FOR RESIDUE 3TR A 1385
ChainResidue
AHOH2360
ALYS273
ASER277
AGLY341
AILE345

site_idAC3
Number of Residues6
DetailsBINDING SITE FOR RESIDUE 3TR B 1386
ChainResidue
BLYS273
BSER277
BGLY341
BILE345
BHOH2346
BHOH2444

site_idAC4
Number of Residues7
DetailsBINDING SITE FOR RESIDUE 3TR A 1386
ChainResidue
ATYR149
APHE207
AASP208
AALA225
AGLY226
AHOH2299
AHOH2300

Functional Information from PROSITE/UniProt
site_idPS00297
Number of Residues8
DetailsHSP70_1 Heat shock hsp70 proteins family signature 1. IDLGTTyS
ChainResidueDetails
AILE9-SER16

site_idPS00329
Number of Residues14
DetailsHSP70_2 Heat shock hsp70 proteins family signature 2. IFDLGGGTfdvSIL
ChainResidueDetails
AILE199-LEU212

site_idPS01036
Number of Residues15
DetailsHSP70_3 Heat shock hsp70 proteins family signature 3. IvLvGGsTRIPkIqK
ChainResidueDetails
AILE336-LYS350

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues10
DetailsBINDING:
ChainResidueDetails
AGLY12
BGLY341
ALYS71
AGLY204
AGLU270
AGLY341
BGLY12
BLYS71
BGLY204
BGLU270

223532

PDB entries from 2024-08-07

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