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5F36

Crystal structure of the bromodomain of human ATAD2 in complex with Compound A12

Functional Information from GO Data
ChainGOidnamespacecontents
A0006325biological_processchromatin organization
A0006355biological_processregulation of transcription, DNA-templated
A0016887molecular_functionATP hydrolysis activity
Functional Information from PDB Data
site_idAC1
Number of Residues6
Detailsbinding site for residue 5UE A 1201
ChainResidue
AALA1060
ATYR1063
AASN1064
AASP1071
AILE1074
AHOH1308

site_idAC2
Number of Residues6
Detailsbinding site for residue SO4 A 1202
ChainResidue
AARG1067
AARG1072
AHOH1355
AARG987
AARG990
AARG994

site_idAC3
Number of Residues1
Detailsbinding site for residue CL A 1203
ChainResidue
AARG1077

222415

PDB entries from 2024-07-10

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