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5F04

Structure of Transcriptional Regulatory Repressor Protein - EthR from Mycobacterium Tuberculosis in complex with compound 3 at 1.84A resolution

Functional Information from GO Data
ChainGOidnamespacecontents
A0000976molecular_functiontranscription cis-regulatory region binding
A0003677molecular_functionDNA binding
A0003700molecular_functionDNA-binding transcription factor activity
A0005515molecular_functionprotein binding
A0005829cellular_componentcytosol
A0006355biological_processregulation of DNA-templated transcription
A0045892biological_processnegative regulation of DNA-templated transcription
A0046677biological_processresponse to antibiotic
Functional Information from PDB Data
site_idAC1
Number of Residues14
Detailsbinding site for residue 5TB A 301
ChainResidue
APHE110
AASN179
AGLU180
ALEU183
APHE184
ATRP207
APHE114
ATHR121
AGLN125
AMET142
ATRP145
ATYR148
ATHR149
AASN176

site_idAC2
Number of Residues3
Detailsbinding site for residue SO4 A 302
ChainResidue
AASP98
AARG99
AHOH403

site_idAC3
Number of Residues3
Detailsbinding site for residue SO4 A 303
ChainResidue
AMET102
ATRP103
AVAL152

site_idAC4
Number of Residues6
Detailsbinding site for residue GOL A 304
ChainResidue
AASP154
AARG157
AARG164
AARG164
APRO167
AALA168

site_idAC5
Number of Residues5
Detailsbinding site for residue EDO A 305
ChainResidue
APRO41
ALEU42
AARG122
AALA123
AHOH407

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues19
DetailsDNA_BIND: H-T-H motif => ECO:0000255|PROSITE-ProRule:PRU00335
ChainResidueDetails
ASER46-PHE65

site_idSWS_FT_FI2
Number of Residues2
DetailsSITE: Inhibitor-binding
ChainResidueDetails
AASN176
AASN179

222415

PDB entries from 2024-07-10

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