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5EU8

Structure of FIPV main protease in complex with dual inhibitors

Functional Information from GO Data
ChainGOidnamespacecontents
A0008233molecular_functionpeptidase activity
A0019082biological_processviral protein processing
Functional Information from PDB Data
site_idAC1
Number of Residues4
DetailsBINDING SITE FOR RESIDUE ZN A 401
ChainResidue
AHIS41
AHIS163
AASP186
AHOH558

site_idAC2
Number of Residues4
DetailsBINDING SITE FOR RESIDUE EDO A 402
ChainResidue
ASER104
AGLU179
AHOH532
AHOH532

site_idAC3
Number of Residues16
DetailsBINDING SITE FOR CHAIN B OF N-[(5-METHYLISOXAZOL-3-YL)CARBONYL]ALANYL-L-VALYL-N~1~-((1R,2Z)-4-(BENZYLOXY)-4-OXO-1-{[(3R)-2-OXOPYRROLIDIN-3-YL]METHYL}BUT-2-ENYL)-L-LEUCINAMIDE
ChainResidue
AVAL26
AHIS41
ACYS144
AHIS162
AHIS163
ALEU164
AGLU165
AGLY167
AGLN187
APRO188
ASER189
AMET190
AALA252
ALYS253
AHOH574
AASN25

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues2
DetailsActive site: {"description":"For 3CL-PRO activity"}
ChainResidueDetails

site_idSWS_FT_FI2
Number of Residues1
DetailsSite: {"description":"Important for substrate recognition"}
ChainResidueDetails

239492

PDB entries from 2025-07-30

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