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5EPN

Crystal structure of HCV NS3/4A protease in complex with 5172-mcP1P3 (MK-5172 P1-P3 macrocyclic analogue)

Functional Information from GO Data
ChainGOidnamespacecontents
A0003724molecular_functionRNA helicase activity
A0004252molecular_functionserine-type endopeptidase activity
A0006508biological_processproteolysis
A0008233molecular_functionpeptidase activity
A0008236molecular_functionserine-type peptidase activity
A0008270molecular_functionzinc ion binding
A0016787molecular_functionhydrolase activity
A0019062biological_processvirion attachment to host cell
A0019087biological_processsymbiont-mediated transformation of host cell
A0033644cellular_componenthost cell membrane
A0039502biological_processsymbiont-mediated suppression of host type I interferon-mediated signaling pathway
A0039545biological_processsymbiont-mediated suppression of host cytoplasmic pattern recognition receptor signaling pathway via inhibition of MAVS activity
A0043657cellular_componenthost cell
A0046718biological_processsymbiont entry into host cell
A0046872molecular_functionmetal ion binding
A0052031biological_processsymbiont-mediated perturbation of host defense response
A0052170biological_processsymbiont-mediated suppression of host innate immune response
A0055036cellular_componentvirion membrane
Functional Information from PDB Data
site_idAC1
Number of Residues4
Detailsbinding site for residue ZN A 1201
ChainResidue
ACYS1097
ACYS1099
ACYS1145
AHIS1149

site_idAC2
Number of Residues8
Detailsbinding site for residue SO4 A 1202
ChainResidue
AHOH1336
AHOH1359
AHOH1379
ATYR1006
AGLN1008
ATYR1056
A5R21203
AHOH1311

site_idAC3
Number of Residues20
Detailsbinding site for residue 5R2 A 1203
ChainResidue
APHE1043
ATYR1056
AHIS1057
AGLY1058
AVAL1078
AASP1081
AILE1132
ALEU1135
ALYS1136
AGLY1137
ASER1138
ASER1139
APHE1154
AARG1155
AALA1156
AALA1157
ASO41202
AHOH1321
AHOH1350
AHOH1351

257179

PDB entries from 2026-07-29

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