5DYB
Crystal Structure of the ER-alpha Ligand-binding Domain in Complex with the Cyclofenil Derivative 4,4'-(3,4-dihydronaphthalen-2(1H)-ylidenemethanediyl)diphenol
Functional Information from PDB Data
site_id | AC1 |
Number of Residues | 12 |
Details | binding site for residue 5K2 A 900 |
Chain | Residue |
A | MET343 |
A | LEU428 |
A | LEU525 |
A | LEU540 |
A | LEU346 |
A | THR347 |
A | ALA350 |
A | GLU353 |
A | LEU387 |
A | ARG394 |
A | MET421 |
A | ILE424 |
site_id | AC2 |
Number of Residues | 12 |
Details | binding site for residue 5K2 B 901 |
Chain | Residue |
B | LEU346 |
B | THR347 |
B | ALA350 |
B | GLU353 |
B | LEU387 |
B | ARG394 |
B | PHE404 |
B | MET421 |
B | ILE424 |
B | PHE425 |
B | LEU428 |
B | LEU540 |
Functional Information from SwissProt/UniProt
site_id | SWS_FT_FI1 |
Number of Residues | 2 |
Details | MOD_RES: Phosphoserine => ECO:0007744|PubMed:23186163, ECO:0007744|PubMed:24275569 |
Chain | Residue | Details |
C | SER699 | |
D | SER699 |
site_id | SWS_FT_FI2 |
Number of Residues | 2 |
Details | LIPID: S-palmitoyl cysteine => ECO:0000250 |
Chain | Residue | Details |
A | CYS447 | |
B | CYS447 |