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5DV8

Human PPARgamma ligand binding dmain complexed with SB1451 in a covalent bonded form

Functional Information from GO Data
ChainGOidnamespacecontents
A0003677molecular_functionDNA binding
A0004879molecular_functionnuclear receptor activity
A0005634cellular_componentnucleus
A0006355biological_processregulation of DNA-templated transcription
Functional Information from PDB Data
site_idAC1
Number of Residues19
Detailsbinding site for residue T51 A 501
ChainResidue
AILE262
AARG288
ASER289
AILE326
AILE341
ASER342
AGLU351
APHE363
ALEU465
ALEU469
ATYR473
ALYS263
ALYS265
AHIS266
APHE282
AGLY284
ACYS285
AGLN286
APHE287

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues1
DetailsMOD_RES: Phosphoserine => ECO:0007744|PubMed:23186163
ChainResidueDetails
BSER698
AHIS323
AHIS449
ATYR473

site_idSWS_FT_FI2
Number of Residues2
DetailsCROSSLNK: Glycyl lysine isopeptide (Lys-Gly) (interchain with G-Cter in ubiquitin) => ECO:0000269|PubMed:36737649
ChainResidueDetails
ALYS224

237423

PDB entries from 2025-06-11

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