Loading
PDBj
MenuPDBj@FacebookPDBj@TwitterPDBj@YouTubewwPDB FoundationwwPDB
RCSB PDBPDBeBMRBAdv. SearchSearch help

5DFC

Crystal structure of BRD2(BD2) W370F mutant with ligand I-BET 762 bound

Functional Information from PDB Data
site_idAC1
Number of Residues7
Detailsbinding site for residue GOL A 501
ChainResidue
ATYR368
ALYS402
AASP407
AMET438
ALYS441
AHOH605
AHOH641

site_idAC2
Number of Residues8
Detailsbinding site for residue 2PE A 502
ChainResidue
AASP385
AGLU404
ATYR428
AASN429
AEAM503
AHOH650
ASER347
ALYS351

site_idAC3
Number of Residues9
Detailsbinding site for residue EAM A 503
ChainResidue
APRO371
ALEU383
AASN429
AVAL435
AMET438
A2PE502
AHOH606
AHOH611
AHOH626

site_idAC4
Number of Residues4
Detailsbinding site for residue NI A 504
ChainResidue
AARG419
AARG419
AHOH637
AHOH637

Functional Information from PROSITE/UniProt
site_idPS00633
Number of Residues60
DetailsBROMODOMAIN_1 Bromodomain signature. AfpFykpvDasalglhDYHdiIkhpMdlstVkrkmenrd..Yrdaqefaadvrl.MfsNCykY
ChainResidueDetails
AALA369-TYR428

224201

PDB entries from 2024-08-28

PDB statisticsPDBj update infoContact PDBjnumon