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5DDE

Menin in complex with MI-859

Functional Information from GO Data
ChainGOidnamespacecontents
A0005634cellular_componentnucleus
Functional Information from PDB Data
site_idAC1
Number of Residues19
Detailsbinding site for residue 5A0 A 601
ChainResidue
ASER155
AMET278
AASN282
ATYR319
AMET322
ATYR323
A5A0602
ADMS607
ADMS608
AHOH814
AHOH990
ALEU177
ASER178
AASP180
AHIS181
AALA182
APHE238
ACYS241
ATYR276

site_idAC2
Number of Residues15
Detailsbinding site for residue 5A0 A 602
ChainResidue
ASER155
ALEU177
ASER178
APHE238
ACYS241
ATYR276
AMET278
AASN282
ATYR319
AMET322
ATYR323
A5A0601
ADMS607
ADMS608
AHOH814

site_idAC3
Number of Residues7
Detailsbinding site for residue SO4 A 603
ChainResidue
AARG332
AVAL334
AARG335
AGLY401
AALA403
AHOH873
AHOH895

site_idAC4
Number of Residues3
Detailsbinding site for residue SO4 A 604
ChainResidue
APRO12
AARG14
AHOH705

site_idAC5
Number of Residues4
Detailsbinding site for residue SO4 A 605
ChainResidue
ALYS377
AARG446
AHOH919
AHOH960

site_idAC6
Number of Residues4
Detailsbinding site for residue SO4 A 606
ChainResidue
ATYR133
APHE134
AARG137
AARG332

site_idAC7
Number of Residues4
Detailsbinding site for residue DMS A 607
ChainResidue
ASER155
A5A0601
A5A0602
ADMS608

site_idAC8
Number of Residues6
Detailsbinding site for residue DMS A 608
ChainResidue
ASER155
APHE238
AALA242
A5A0601
A5A0602
ADMS607

site_idAC9
Number of Residues6
Detailsbinding site for residue DMS A 609
ChainResidue
APHE43
APHE47
AGLY386
AGLN400
AHOH723
AHOH947

site_idAD1
Number of Residues6
Detailsbinding site for residue PG4 A 610
ChainResidue
ALEU75
ATHR76
APHE365
AHOH799
AHOH975
AHOH981

site_idAD2
Number of Residues4
Detailsbinding site for residue DMS A 611
ChainResidue
AGLY190
AGLU191
AARG229
ASER583

site_idAD3
Number of Residues2
Detailsbinding site for residue EDO A 612
ChainResidue
ATRP126
ALYS135

238895

PDB entries from 2025-07-16

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